SCHEMBL9437769

SCHEMBL9437769

O=C1COc2ccc(CCNCCCCN3CCCCC3=O)cc2N1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.47
NR3C2 P08235 1/20 0.44
HTR1A P08908 9/20 0.43
DRD2 P14416 5/20 0.43
HTR2A P28223 3/20 0.43
HTR1D P28221 6/20 0.43
HTR1B P28222 6/20 0.43
SLC6A4 P31645 4/20 0.43
DRD4 P21917 3/20 0.42
DRD3 P35462 2/20 0.42
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9437890 0.85 HTR1A (0.47) PARP1NR3C2HTR1ADRD2HTR2A
SCHEMBL9437874 0.80 PARP1 (0.49) PARP1NR3C2HTR1ADRD2HTR2A
SCHEMBL9437900 0.80 PARP1 (0.46) PARP1NR3C2HTR1ADRD2HTR2A
SCHEMBL9437866 0.79 PARP1 (0.53) PARP1NR3C2HTR1ADRD2HTR2A
SCHEMBL9452085 0.79 HTR1A (0.47) HTR1ADRD2HTR2AHTR1DHTR1B
SCHEMBL9437815 0.79 PARP1 (0.45) PARP1NR3C2HTR1ADRD2HTR2A
SCHEMBL9437714 0.76 PARP1 (0.67) PARP1NR3C2HTR1ADRD2HTR1D
SCHEMBL9437847 0.76 PARP1 (0.54) PARP1NR3C2HTR1ADRD2HTR2A
SCHEMBL9437965 0.75 HTR1A (0.52) HTR1AHTR1DHTR1BSLC6A4DRD4
SCHEMBL9437860 0.73 PARP1 (0.56) PARP1NR3C2HTR1ADRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5196434-A Antidepressants, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-03-23 US disclosed
EP-0478446-A1 Heterocyclic alkylamines, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-04-01 EP disclosed