SCHEMBL9437890

SCHEMBL9437890

CC1(C)CCN(CCCCNCCc2ccc3c(c2)NC(=O)CO3)C(=O)C1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.47
HTR1D P28221 8/20 0.47
HTR1B P28222 8/20 0.47
SLC6A4 P31645 6/20 0.47
PARP1 P09874 4/20 0.46
NR3C2 P08235 1/20 0.43
DRD2 P14416 8/20 0.41
HTR2A P28223 3/20 0.41
DRD4 P21917 5/20 0.41
DRD3 P35462 3/20 0.41
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9437874 0.87 PARP1 (0.49) HTR1AHTR1DHTR1BSLC6A4PARP1
SCHEMBL9437769 0.85 PARP1 (0.47) HTR1AHTR1DHTR1BSLC6A4PARP1
SCHEMBL9437887 0.83 HTR1A (0.45) HTR1AHTR1DHTR1BSLC6A4DRD2
SCHEMBL9437802 0.79 HTR1A (0.49) HTR1AHTR1DHTR1BSLC6A4DRD2
SCHEMBL9437815 0.78 PARP1 (0.45) HTR1AHTR1DHTR1BSLC6A4PARP1
SCHEMBL9437866 0.76 PARP1 (0.53) HTR1AHTR1DHTR1BSLC6A4PARP1
SCHEMBL9437714 0.76 PARP1 (0.67) HTR1AHTR1DHTR1BSLC6A4PARP1
SCHEMBL9437900 0.75 PARP1 (0.46) HTR1AHTR1DHTR1BSLC6A4PARP1
SCHEMBL9437800 0.74 SIGMAR1 (0.46) HTR1AHTR2C
SCHEMBL9437794 0.74 HTR1A (0.46) HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5268381-A Antidepressant or anxiolytic compound ADIR ET COMPAGNIE (FR) 1993-12-07 US disclosed
US-5242772-A Process for the production of a lithographic printing plate of direct image type FUJI PHOTO FILM CO., LTD. (JP) 1993-09-07 US disclosed
US-5196434-A Antidepressants, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-03-23 US disclosed