SCHEMBL9437815

SCHEMBL9437815

O=C1COc2ccc(CCNCCCCN3C(=O)CC4(CCCCC4)C3=O)cc2N1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.45
NR3C2 P08235 3/20 0.41
HTR1A P08908 8/20 0.41
HTR1B P28222 6/20 0.41
HTR1D P28221 5/20 0.41
SLC6A4 P31645 4/20 0.41
DRD2 P14416 4/20 0.39
HTR2A P28223 3/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
DRD1 P21728 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9437874 0.84 PARP1 (0.49) PARP1NR3C2HTR1AHTR1BHTR1D
SCHEMBL9437710 0.82 HTR1A (0.42) HTR1AHTR1BHTR1DSLC6A4DRD2
SCHEMBL9437886 0.82 PARP1 (0.44) PARP1NR3C2HTR1AHTR1BHTR1D
SCHEMBL9437900 0.80 PARP1 (0.46) PARP1NR3C2HTR1AHTR1BHTR1D
SCHEMBL9437866 0.79 PARP1 (0.53) PARP1NR3C2HTR1AHTR1BHTR1D
SCHEMBL9437769 0.79 PARP1 (0.47) PARP1NR3C2HTR1AHTR1BHTR1D
SCHEMBL9437808 0.79 HTR1A (0.45) HTR1AHTR1BHTR1DSLC6A4DRD2
SCHEMBL9437890 0.78 HTR1A (0.47) PARP1NR3C2HTR1AHTR1BHTR1D
SCHEMBL9437847 0.76 PARP1 (0.54) PARP1NR3C2HTR1AHTR1BHTR1D
SCHEMBL9437929 0.74 HTR1A (0.43) HTR1ASLC6A4CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5268381-A Antidepressant or anxiolytic compound ADIR ET COMPAGNIE (FR) 1993-12-07 US disclosed