SCHEMBL9440341

SCHEMBL9440341

OC(c1ccc(F)cc1)c1ccc(I)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.42
NR3C1 P04150 1/20 0.40
APP P05067 1/20 0.39
AOC3 Q16853 1/20 0.38
IDO1 P14902 2/20 0.38
TDO2 P48775 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.36
BRD4 O60885 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14160109 0.87 CYP17A1 (0.38) SMN1; SMN2
SCHEMBL597442 0.87 IDO1 (0.46) NR3C1AOC3IDO1TDO2HDAC3
SCHEMBL7079520 0.80 NR3C1 (0.42) NR3C1AOC3IDO1TDO2HDAC3
SCHEMBL18472615 0.79
SCHEMBL1216 0.79
SCHEMBL24238297 0.78 SMN1; SMN2 (0.48) KMT2AKDM4ELMNASMN1; SMN2
SCHEMBL21542545 0.78 EPHX1 (0.48) NR3C1KMT2AATMKDM4EALDH1A1
SCHEMBL21542539 0.78 EPHX1 (0.48) NR3C1KMT2AATMKDM4EALDH1A1
SCHEMBL477477 0.78 EPHX1 (0.48) NR3C1KMT2AATMKDM4EALDH1A1
SCHEMBL9440465 0.78 CYP3A4 (0.52) APPKMT2AKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276037-A Antiinflammatory agents, antiallergens IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-01-04 US disclosed
US-5272173-A 5-lipoxygenase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-21 US disclosed
US-5225438-A Lipoxygenase inhibitors for antiinflammatory agents or antiallergens IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-07-06 US disclosed
EP-0488602-A1 Aryl derivatives ZENECA LIMITED (GB) 1992-06-03 EP disclosed
EP-0485111-A2 The use of lipoxygenase and cyclooxygenase inhibitors as synergistic agents ZENECA LIMITED (GB) 1992-05-13 EP disclosed