SCHEMBL9440384

SCHEMBL9440384

Nc1ccc(Oc2ccc(Br)cc2Cl)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.57
PDE7A Q13946 2/20 0.56
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
ALDH1A1 P00352 6/20 0.45
CYP3A4 P08684 1/20 0.45
TSHR P16473 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
KDM4E B2RXH2 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTR2A P28223 2/20 0.42
SLC6A4 P31645 2/20 0.42
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22069698 0.89 MAPT (0.57) MAPTPDE7AMAOAMAOBALDH1A1
SCHEMBL9272342 0.85 MAPT (0.50) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL4318630 0.85 PDE7A (0.63) MAPTPDE7AMAOAMAOBALDH1A1
SCHEMBL10962941 0.83 MAPT (0.55) MAPTPDE7AALDH1A1CYP3A4TSHR
SCHEMBL8683893 0.82 STK39 (0.46) MAPTTSHRMEN1KMT2AHPGD
SCHEMBL9440387 0.82 SCN9A (0.44) PDE7AALDH1A1TDP1HTR2ASLC6A4
SCHEMBL11606863 0.82 MAPT (0.47) MAPTALDH1A1TSHRTDP1MEN1
SCHEMBL8683891 0.82 KMT2A (0.43) MAPTPDE7AALDH1A1TSHRTDP1
SCHEMBL1129611 0.81 SLC6A4 (0.50) MAPTALDH1A1CYP3A4TSHRTDP1
SCHEMBL554810 0.81 MAOA (0.61) MAPTPDE7AMAOAMAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276037-A Antiinflammatory agents, antiallergens IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-01-04 US disclosed
US-5272173-A 5-lipoxygenase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-21 US disclosed
US-5225438-A Lipoxygenase inhibitors for antiinflammatory agents or antiallergens IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-07-06 US disclosed
EP-0488602-A1 Aryl derivatives ZENECA LIMITED (GB) 1992-06-03 EP disclosed
US-4355186-A Process for the preparation of 4-phenoxy-phenols HOECHST AKTIENGESELLSCHAFT (DE) 1982-10-19 US disclosed