SCHEMBL9440464

SCHEMBL9440464

FC(F)(F)c1ccc(Cc2ccc(I)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.50
TAAR1 Q96RJ0 1/20 0.48
IDO1 P14902 4/20 0.47
TRPV1 Q8NER1 1/20 0.46
LTA4H P09960 1/20 0.45
MAOB P27338 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KIF11 P52732 1/20 0.40
KMT2A Q03164 1/20 0.40
MIF P14174 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
IDH1 O75874 1/20 0.39
APP P05067 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2096666 0.88 SRD5A2 (0.59) SRD5A2TAAR1IDO1LTA4HMAOB
SCHEMBL1616 0.85 TRPV1 (0.55) TAAR1IDO1TRPV1ALDH1A1KIF11
SCHEMBL25191871 0.83 TRPV1 (0.53) TAAR1IDO1TRPV1ALDH1A1KIF11
Phosphine SCHEMBL28192244 0.83 TRPV1 (0.53) TAAR1IDO1TRPV1ALDH1A1KIF11
SCHEMBL5491719 0.80 CYP3A4 (0.50) IDO1ALDH1A1APP
SCHEMBL5255445 0.79 ALDH1A1 (0.59) SRD5A2TAAR1IDO1LTA4HMAOB
SCHEMBL7935401 0.79 SRD5A2 (0.52) SRD5A2TAAR1IDO1LTA4HMAOB
SCHEMBL6547427 0.78 KIF11 (0.61) TRPV1MAOBALDH1A1KIF11
SCHEMBL5695842 0.78 TRPV1 (0.50) TAAR1TRPV1ALDH1A1KIF11KMT2A
SCHEMBL5511243 0.77 SRD5A2 (0.50) SRD5A2TAAR1IDO1LTA4HMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276037-A Antiinflammatory agents, antiallergens IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-01-04 US disclosed
US-5272173-A 5-lipoxygenase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-21 US disclosed
US-5225438-A Lipoxygenase inhibitors for antiinflammatory agents or antiallergens IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-07-06 US disclosed
EP-0488602-A1 Aryl derivatives ZENECA LIMITED (GB) 1992-06-03 EP disclosed