SCHEMBL9440635

SCHEMBL9440635

c1ccc(CCOc2ccccc2OC(CC2=NCCN2)c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 14/20 0.51
MAOA P21397 7/20 0.49
MAOB P27338 7/20 0.49
ADRA2A P08913 5/20 0.44
ADRA2B P18089 5/20 0.44
ADRA2C P18825 5/20 0.44
ADRA1A P35348 3/20 0.44
TAAR1 Q96RJ0 2/20 0.44
ADRA1D P25100 2/20 0.44
ADRA1B P35368 2/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
TSHR P16473 1/20 0.44
HTR1A P08908 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7854312 0.81 ADRA2B (0.50) NISCHMAOAMAOBADRA2AADRA2B
SCHEMBL9440693 0.81 NISCH (0.52) NISCHMAOAMAOBADRA2AADRA2B
SCHEMBL9440600 0.81 NISCH (0.52) NISCHMAOAMAOBADRA2AADRA2B
SCHEMBL9440508 0.80 NISCH (0.53) NISCHMAOAMAOBADRA2AADRA2B
SCHEMBL9440279 0.80 NISCH (0.57) NISCHMAOAMAOBADRA2AADRA2B
SCHEMBL9440611 0.77 NISCH (0.50) NISCHMAOAMAOBADRA2AADRA2B
SCHEMBL9445174 0.75 NISCH (0.55) NISCHMAOAMAOBADRA2AADRA2B
SCHEMBL9201353 0.70 ADRA2A (0.66) NISCHMAOAMAOBADRA2AADRA2B
SCHEMBL7547171 0.70 NISCH (1.00) NISCHMAOAMAOBADRA2AADRA2B
SCHEMBL3169171 0.69 NISCH (0.52) NISCHMAOAMAOBADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625969-A1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL PHARMACEUTICALS INC. (US) 1994-11-30 EP claimed