SCHEMBL9447237

SCHEMBL9447237

O=C1COSc2ccccc2-c2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
MAOA P21397 3/20 0.35
MAOB P27338 2/20 0.35
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
S100A4 P26447 3/20 0.34
BLM P54132 2/20 0.34
BCHE P06276 2/20 0.34
CES1 P23141 2/20 0.34
POLB P06746 2/20 0.34
CES2 O00748 1/20 0.34
APAF1 O14727 1/20 0.34
TERT O14746 1/20 0.34
NPC1 O15118 1/20 0.34
PLIN1 O60240 1/20 0.34
TDP2 O95551 1/20 0.34
S1PR4 O95977 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65679 0.69 MAOB (0.42) KDM4EALDH1A1HPGDMAOAMAOB
SCHEMBL5281409 0.66
SCHEMBL31218602 0.66 MAOA (0.60) KDM4EALDH1A1HPGDMAOAMAOB
SCHEMBL7380169 0.66 MAOA (0.60) KDM4EALDH1A1HPGDMAOAMAOB
SCHEMBL2929432 0.65 PKM (0.52) KDM4EALDH1A1HPGDMAOAMAOB
SCHEMBL1913191 0.64 BRD4 (0.47) ALDH1A1MAOAMEN1KMT2ABCHE
SCHEMBL10556518 0.64 MAOA (0.53) KDM4EALDH1A1HPGDMAOAMAOB
SCHEMBL855431 0.61 MAOA (0.56) KDM4EMAOAMAOBMEN1KMT2A
SCHEMBL19537629 0.61 ALDH1A1 (0.48) KDM4EALDH1A1HPGDMAOAMEN1
SCHEMBL88188 0.61 CES1 (0.52) KDM4EALDH1A1HPGDMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0490219-A1 Substituted dibenz-oxo-thiocinones, -12-oxides and -12,12-dioxides; method for their preparation and their use in medicaments BAYER AG (DE) 1992-06-17 EP claimed
US-5190971-A SUBSTITUTED DIBENZ-OXA-THIOCINONES, -12-OXIDES AND -12,12-DIOXIDES, A PROCESS FOR THEIR PREPARATION AND THEIR USE IN MEDICAMENTS BAYER AKTIENGESELLSCHAFT (DE) 1993-03-02 US disclosed
EP-0490219-A1 Substituted dibenz-oxo-thiocinones, -12-oxides and -12,12-dioxides; method for their preparation and their use in medicaments BAYER AG (DE) 1992-06-17 EP disclosed
EP-0490219-A1 Substituted dibenz-oxo-thiocinones, -12-oxides and -12,12-dioxides; method for their preparation and their use in medicaments BAYER AG (DE) 1992-06-17 EP disclosed