SCHEMBL9449122

SCHEMBL9449122

CC(=O)Oc1ccc2[nH]cc(C3CN4CCC3CC4)c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.50
MTNR1B P49286 1/20 0.50
NOS3 P29474 3/20 0.48
NOS1 P29475 3/20 0.48
HTR1D P28221 4/20 0.46
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
HTR1B P28222 3/20 0.43
HTR1A P08908 2/20 0.43
HTR1F P30939 1/20 0.43
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNA7 P36544 1/20 0.42
CHRNA4 P43681 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9448887 0.91 NOS3 (0.48) MTNR1AMTNR1BNOS3NOS1HTR1D
SCHEMBL9448764 0.88 HTR1B (0.49) MTNR1AMTNR1BNOS3NOS1HTR1D
SCHEMBL9449079 0.88 HTR1D (0.47) MTNR1AMTNR1BNOS3NOS1HTR1D
SCHEMBL9449276 0.87 NOS3 (0.46) MTNR1AMTNR1BNOS3NOS1HTR1D
SCHEMBL9448836 0.85 HTR2A (0.61) MTNR1AMTNR1BNOS3NOS1HTR2A
SCHEMBL9449214 0.82 NOS3 (0.46) MTNR1AMTNR1BNOS3NOS1HTR1D
SCHEMBL9448957 0.82 NOS3 (0.48) MTNR1AMTNR1BNOS3NOS1HTR1D
SCHEMBL9449109 0.80 HTR1A (0.47) MTNR1AMTNR1BNOS3NOS1HTR1D
SCHEMBL9448885 0.80 NOS3 (0.46) MTNR1AMTNR1BNOS3NOS1HTR1D
SCHEMBL9449161 0.80 NOS3 (0.46) MTNR1AMTNR1BNOS3NOS1HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5227386-A INDOLE DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-07-13 US disclosed