SCHEMBL9449161

SCHEMBL9449161

CC(C)(C)C(=O)Oc1ccc2c(C3CN4CCC3CC4)c[nH]c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.46
NOS1 P29475 3/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
NOS2 P35228 1/20 0.46
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
GABRA1 P14867 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
HSD11B1 P28845 1/20 0.37
KDM4E B2RXH2 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9449079 0.92 HTR1D (0.47) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448887 0.88 NOS3 (0.48) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448885 0.85 NOS3 (0.46) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448872 0.82 NOS3 (0.49) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9449086 0.80 GABRA1 (0.41) HTR1DHTR1BGABRA1GABRG2GABRB3
SCHEMBL9449122 0.80 MTNR1A (0.50) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448798 0.80 NOS3 (0.46) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448897 0.78 NOS3 (0.54) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448764 0.77 HTR1B (0.49) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9449276 0.76 NOS3 (0.46) NOS3NOS1CYP3A4CYP2C19NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5227386-A INDOLE DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-07-13 US disclosed