SCHEMBL9449079

SCHEMBL9449079

CC(C)(C)C(=O)Oc1ccc2[nH]cc(C3CN4CCC3CC4)c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 4/20 0.47
HTR1B P28222 4/20 0.47
NOS3 P29474 3/20 0.46
NOS1 P29475 3/20 0.46
MTNR1A P48039 1/20 0.45
MTNR1B P49286 1/20 0.45
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 1/20 0.40
NOS2 P35228 1/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNA4 P43681 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9449161 0.92 NOS3 (0.46) HTR1DHTR1BNOS3NOS1MTNR1A
SCHEMBL9449122 0.88 MTNR1A (0.50) HTR1DHTR1BNOS3NOS1MTNR1A
SCHEMBL9448764 0.85 HTR1B (0.49) HTR1DHTR1BNOS3NOS1MTNR1A
SCHEMBL9449276 0.84 NOS3 (0.46) HTR1DHTR1BNOS3NOS1MTNR1A
SCHEMBL9448836 0.82 HTR2A (0.61) HTR1BNOS3NOS1MTNR1AMTNR1B
SCHEMBL9449136 0.80 LMNA (0.38) HTR1DHTR1BMTNR1AMTNR1B
SCHEMBL9448887 0.80 NOS3 (0.48) HTR1DHTR1BNOS3NOS1MTNR1A
SCHEMBL9449214 0.80 NOS3 (0.46) HTR1DHTR1BNOS3NOS1MTNR1A
SCHEMBL9448957 0.79 NOS3 (0.48) HTR1DHTR1BNOS3NOS1MTNR1A
SCHEMBL3546179 0.78 CYP3A4 (0.56) HTR1DHTR1BNOS3NOS1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5227386-A INDOLE DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-07-13 US disclosed