SCHEMBL9449953

SCHEMBL9449953

O=C(O)COc1cc[c]cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.56
TSHR P16473 1/20 0.50
CYP2C19 P33261 1/20 0.49
KMT2A Q03164 1/20 0.47
PTGDR2 Q9Y5Y4 7/20 0.45
MAPT P10636 1/20 0.44
POLB P06746 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GLA P06280 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MCL1 Q07820 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
CASP1 P29466 1/20 0.40
PPARG P37231 1/20 0.40
CASP7 P55210 1/20 0.40
NCOA2 Q15596 1/20 0.40
NCOA1 Q15788 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2317153 0.86 TDP1 (0.51) TDP1TSHRCYP2C19KMT2APTGDR2
SCHEMBL6718467 0.84 L3MBTL1 (0.50) TDP1TSHRKMT2APTGDR2MAPT
SCHEMBL9449849 0.82 LMNA (0.55) TDP1TSHRKMT2APTGDR2MAPT
SCHEMBL9449949 0.80 ALDH1A1 (0.46) TDP1TSHRKMT2AL3MBTL1KDM4E
SCHEMBL3931134 0.79 PKM (0.45) TDP1PTGDR2POLBSMN1; SMN2GLA
SCHEMBL5619089 0.79 KDM4E (0.44) TDP1CYP2C19KMT2APTGDR2POLB
SCHEMBL5503687 0.79 PKM (0.53) TDP1TSHRPTGDR2POLBSMN1; SMN2
SCHEMBL7380176 0.78 POLB (0.62) TDP1TSHRKMT2APTGDR2POLB
SCHEMBL3209384 0.78 POLB (0.62) TDP1TSHRKMT2APTGDR2POLB
SCHEMBL5460045 0.77 L3MBTL1 (0.65) TDP1TSHRKMT2APTGDR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5232978-A 1-(2-arylethyl)-pyrrolidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-08-03 US disclosed
EP-0483580-A2 1-(2-Arylethyl)-pyrrolidine MERCK PATENT GmbH (DE) 1992-05-06 EP disclosed
EP-0374756-A2 Nitrogen-containing cyclic compounds MERCK PATENT GmbH (DE) 1990-06-27 EP disclosed