SCHEMBL945358

SCHEMBL945358

CC1=NC(C)(c2cccc(Br)c2)N=C1N

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 14/20 0.58
KCNH2 Q12809 1/20 0.58
APP P05067 6/20 0.43
CTSD P07339 1/20 0.41
DHFR P00374 1/20 0.38
HTR1A P08908 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR7 P34969 1/20 0.38
HTR2B P41595 1/20 0.38
HTR5A P47898 1/20 0.38
HTR6 P50406 1/20 0.38
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
CHRNA1 P02708 1/20 0.37
CHRNG P07510 1/20 0.37
CHRNB1 P11230 1/20 0.37
CHRNB2 P17787 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931186 0.81 CHRNA1 (0.40) BACE1KCNH2CTSDDHFRHTR1A
SCHEMBL932046 0.78 BACE1 (0.60) BACE1KCNH2APPCTSD
SCHEMBL932309 0.78 BACE1 (0.44) BACE1KCNH2APPCTSDDHFR
SCHEMBL932262 0.77 BACE1 (0.40) BACE1KCNH2APPCTSDDHFR
SCHEMBL932108 0.75 BACE1 (0.62) BACE1KCNH2APPCTSD
SCHEMBL932230 0.75 BACE1 (0.59) BACE1KCNH2APP
SCHEMBL932111 0.75 BACE1 (0.47) BACE1KCNH2APPCTSDALDH1A1
SCHEMBL932149 0.74 BACE1 (1.00) BACE1KCNH2
SCHEMBL932138 0.74 BACE1 (1.00) BACE1KCNH2
SCHEMBL6893840 0.74 BACE1 (1.00) BACE1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed