SCHEMBL932309

SCHEMBL932309

CCC1(c2cccc(Br)c2)N=C(C)C(N)=N1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.44
APP P05067 8/20 0.41
KCNH2 Q12809 1/20 0.37
CTSD P07339 1/20 0.37
KDM1A O60341 1/20 0.35
RCOR1 Q9UKL0 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
DHFR P00374 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932777 0.83 BACE1 (0.65) BACE1APPKCNH2CTSD
SCHEMBL932151 0.82 CHRNA1 (0.35) BACE1CTSDKDM1ARCOR1ALDH1A1
SCHEMBL945358 0.78 BACE1 (0.58) BACE1APPKCNH2CTSDALDH1A1
SCHEMBL6894146 0.78 BACE1 (0.56) BACE1APPKCNH2ALDH1A1
SCHEMBL932274 0.77 BACE1 (0.43) BACE1APPKCNH2
SCHEMBL932046 0.76 BACE1 (0.60) BACE1APPKCNH2CTSD
SCHEMBL932353 0.75 BACE1 (0.69) BACE1KCNH2
SCHEMBL932262 0.75 BACE1 (0.40) BACE1APPKCNH2CTSDALDH1A1
SCHEMBL932230 0.72 BACE1 (0.59) BACE1APPKCNH2
SCHEMBL932108 0.72 BACE1 (0.62) BACE1APPKCNH2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed