SCHEMBL9458362

SCHEMBL9458362

CCN(CC)C(=O)COc1cc(N)c(Cl)cc1C(=O)NCC12CCCN(CC1)C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.47
HTR3E A5X5Y0 3/20 0.45
HTR3B O95264 3/20 0.45
HTR3A P46098 3/20 0.45
HTR3D Q70Z44 3/20 0.45
HTR3C Q8WXA8 3/20 0.45
HTR4 Q13639 5/20 0.41
LMNA P02545 2/20 0.41
CYP1A2 P05177 2/20 0.41
ADRA2A P08913 2/20 0.41
HTR2C P28335 2/20 0.41
DRD3 P35462 2/20 0.41
HTR2B P41595 2/20 0.41
KCNH2 Q12809 2/20 0.41
DRD4 P21917 2/20 0.41
SLC22A1 O15245 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MPO P05164 1/20 0.41
CYP2D6 P10635 1/20 0.41
ADRA2C P18825 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458342 0.85 HTR3E (0.62) DRD2HTR3EHTR3BHTR3AHTR3D
SCHEMBL9458047 0.83 HTR3E (0.52) DRD2HTR3EHTR3BHTR3AHTR3D
SCHEMBL9474371 0.83 HTR3E (0.64) DRD2HTR3EHTR3BHTR3AHTR3D
SCHEMBL9458438 0.82 HTR3E (0.46) DRD2HTR3EHTR3BHTR3AHTR3D
SCHEMBL9622432 0.82 DRD2 (0.49) DRD2HTR3EHTR3BHTR3AHTR3D
SCHEMBL9458602 0.81 HTR3E (0.48) DRD2HTR3EHTR3BHTR3AHTR3D
SCHEMBL9458257 0.81 HTR3E (0.48) DRD2HTR3EHTR3BHTR3AHTR3D
SCHEMBL9474052 0.79 HTR3E (0.46) DRD2HTR3EHTR3BHTR3AHTR3D
SCHEMBL9622436 0.72 GAA (0.60) DRD2HTR3EHTR3BHTR3AHTR3D
SCHEMBL9458494 0.72 ALDH1A1 (0.45) DRD2HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5244907-A Treatment of serotonin imbalance, increase in gastric motility, antiemetics, antiarrhythmia agents A. H. ROBINS COMPANY, INCORPORATED (US) 1993-09-14 US disclosed
US-5190953-A 1-azabicyclo(3.2.1.)octan-5-ylmethyl- or 1-azabicyclo(3.3.1) nonan-5-ylmethyl derivatives of carboxamides, thiocarboxamides or esters, thioesters A. H. ROBINS COMPANY, INCORPORATED (US) 1993-03-02 US disclosed