SCHEMBL9458494

SCHEMBL9458494

CCN(CC)C(=O)COc1cc(N)c(Cl)cc1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
KDM4E B2RXH2 3/20 0.45
HPGD P15428 3/20 0.45
HSD17B10 Q99714 2/20 0.45
TSHR P16473 3/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
HTR3A P46098 2/20 0.44
HTR4 Q13639 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
RAB9A P51151 3/20 0.44
NPC1 O15118 2/20 0.44
DRD2 P14416 2/20 0.44
HTR3E A5X5Y0 1/20 0.44
SLC22A1 O15245 1/20 0.44
HTR3B O95264 1/20 0.44
LMNA P02545 1/20 0.44
MPO P05164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9622436 0.87 GAA (0.60) ALDH1A1SMN1; SMN2KDM4EHPGDHSD17B10
SCHEMBL99475 0.84 TSHR (0.53) ALDH1A1SMN1; SMN2KDM4EHSD17B10TSHR
SCHEMBL22987088 0.79 GAA (0.48) ALDH1A1SMN1; SMN2KDM4ETSHRCYP1A2
SCHEMBL9474066 0.77 HTR4 (0.43) ALDH1A1SMN1; SMN2HPGDTSHRCYP1A2
SCHEMBL7367657 0.76 PTPN11 (0.52) TSHRHTR4CYP3A4LMNAADRA2A
SCHEMBL7267139 0.75 GAA (0.50) ALDH1A1SMN1; SMN2TSHRCYP1A2CYP2D6
SCHEMBL99019 0.74 GAA (0.73) ALDH1A1SMN1; SMN2TSHRCYP1A2CYP2D6
SCHEMBL29242370 0.73 GAA (0.50) ALDH1A1SMN1; SMN2KDM4EHPGDHSD17B10
SCHEMBL9458199 0.73 GAA (0.44) ALDH1A1SMN1; SMN2HPGDHSD17B10TSHR
SCHEMBL11167484 0.73 HSD17B10 (0.49) ALDH1A1SMN1; SMN2HPGDHSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5244907-A Treatment of serotonin imbalance, increase in gastric motility, antiemetics, antiarrhythmia agents A. H. ROBINS COMPANY, INCORPORATED (US) 1993-09-14 US disclosed
US-5190953-A 1-azabicyclo(3.2.1.)octan-5-ylmethyl- or 1-azabicyclo(3.3.1) nonan-5-ylmethyl derivatives of carboxamides, thiocarboxamides or esters, thioesters A. H. ROBINS COMPANY, INCORPORATED (US) 1993-03-02 US disclosed
US-5137895-A Antiemetic, anxiolytic, gastric emptying and serotonin modulating activity A. H. ROBINS COMPANY, INCORPORATED (US) 1992-08-11 US disclosed