SCHEMBL9458592

SCHEMBL9458592

CCc1cc([O])c2cc(F)ccc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.43
PLA2G2A P14555 2/20 0.41
CASP3 P42574 1/20 0.41
TYMS P04818 1/20 0.40
PDE10A Q9Y233 2/20 0.39
TSHR P16473 1/20 0.38
ALDH1A1 P00352 3/20 0.38
GAA P10253 2/20 0.38
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
PRNP P04156 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PARP1 P09874 3/20 0.37
TNKS O95271 2/20 0.37
TNKS2 Q9H2K2 2/20 0.37
MPO P05164 1/20 0.37
POLB P06746 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458576 0.80 ESR1 (0.51) ALDH1A1GAAMEN1HPGDKMT2A
SCHEMBL9458485 0.78 KDM4E (0.50) PLA2G2ATSHRALDH1A1GAAMEN1
SCHEMBL9458599 0.78 ALDH1A1 (0.37) TYMSTSHRALDH1A1GAAMEN1
SCHEMBL26317683 0.78 PDE10A (0.53) DHODHPLA2G2APDE10AMEN1KMT2A
SCHEMBL9458614 0.78 TYMS (0.39) DHODHTYMSTSHRALDH1A1GAA
SCHEMBL9273904 0.77 KDM4E (0.47) ALDH1A1GAAMEN1HPGDKMT2A
SCHEMBL9458139 0.75 APP (0.43) TSHRALDH1A1MEN1HPGDKMT2A
SCHEMBL9458481 0.74 CCNE2 (0.44) ALDH1A1POLB
SCHEMBL9458374 0.74 MAPT (0.43) TSHRALDH1A1GAAMEN1HPGD
SCHEMBL9680806 0.74 ALDH1A1 (0.40) TYMSTSHRALDH1A1MEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5245035-A HETEROCYCLIC BORON COMPOUNDS AS INTERMEDIATES FOR ANGIOTENSIN II ANTAGONISTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-09-14 US claimed
EP-0495627-A1 Boron compounds ZENECA LIMITED (GB) 1992-07-22 EP claimed
US-5245035-A HETEROCYCLIC BORON COMPOUNDS AS INTERMEDIATES FOR ANGIOTENSIN II ANTAGONISTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-09-14 US disclosed
EP-0495627-A1 Boron compounds ZENECA LIMITED (GB) 1992-07-22 EP disclosed