SCHEMBL9458481

SCHEMBL9458481

CCc1cc([O])c2cc(NC=O)ccc2n1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 1/20 0.44
CDK4 P11802 1/20 0.44
CCND1 P24385 1/20 0.44
CCNE1 P24864 1/20 0.44
CDK2 P24941 1/20 0.44
MCHR1 Q99705 13/20 0.39
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
ALDH1A1 P00352 1/20 0.33
OPRL1 P41146 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833601 0.78 NPC1 (0.39) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL9458576 0.74 ESR1 (0.51) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL9458592 0.74 DHODH (0.43) POLBALDH1A1
SCHEMBL9458485 0.72 KDM4E (0.50) NPC1POLBALDH1A1
SCHEMBL9458599 0.72 ALDH1A1 (0.37) MCHR1NPC1POLBALDH1A1
SCHEMBL9458614 0.72 TYMS (0.39) CDK2MCHR1NPC1POLBALDH1A1
SCHEMBL9273904 0.72 KDM4E (0.47) NPC1POLBALDH1A1
SCHEMBL9458374 0.69 MAPT (0.43) POLBALDH1A1OPRL1
SCHEMBL9458139 0.67 APP (0.43) ALDH1A1
SCHEMBL9680806 0.66 ALDH1A1 (0.40) MCHR1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5245035-A HETEROCYCLIC BORON COMPOUNDS AS INTERMEDIATES FOR ANGIOTENSIN II ANTAGONISTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-09-14 US claimed
EP-0495627-A1 Boron compounds ZENECA LIMITED (GB) 1992-07-22 EP claimed
US-5245035-A HETEROCYCLIC BORON COMPOUNDS AS INTERMEDIATES FOR ANGIOTENSIN II ANTAGONISTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-09-14 US disclosed
EP-0495627-A1 Boron compounds ZENECA LIMITED (GB) 1992-07-22 EP disclosed