SCHEMBL9458745

SCHEMBL9458745

CCCCCCc1c(-c2ccccc2)c2n(c1/C=C/C(=O)O)CCC2

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 15/20 0.65
PTGS1 P23219 2/20 0.61
PTGES O14684 1/20 0.41
ESR1 P03372 2/20 0.38
ESR2 Q92731 2/20 0.38
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
CASP3 P42574 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458593 1.00 ALOX5 (0.65) ALOX5PTGS1PTGESESR1ESR2
SCHEMBL9458748 0.86 ALOX5 (0.46) ALOX5PTGS1PTGES
SCHEMBL9458579 0.79 ALOX5 (1.00) ALOX5PTGS1PTGES
SCHEMBL9459144 0.78 PTGES (0.53) ALOX5PTGS1PTGES
SCHEMBL9458649 0.75 PTGES (0.44) ALOX5PTGS1PTGES
SCHEMBL9458503 0.74 ALOX5 (0.70) ALOX5PTGS1PTGESNPC1ALDH1A1
SCHEMBL9458836 0.72 ALOX5 (0.70) ALOX5PTGS1PTGES
SCHEMBL9458881 0.70 OXER1 (0.52) ALOX5PTGS1PTGES
SCHEMBL10445135 0.68 ALOX5 (0.52) ALOX5PTGS1PTGESALDH1A1
SCHEMBL9458661 0.68 CYP2D6 (0.39) PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260451-A Enzyme inhibitors MERCKLE GMBH (DE) 1993-11-09 US disclosed
EP-0397175-A1 Substituted pyrrolizine compounds and theit use as pharmaceuticals Dannhardt, Gerd, Prof.Dr. (DE) 1990-11-14 EP disclosed