SCHEMBL9458649

SCHEMBL9458649

CCCCCCc1c(C=O)c(-c2ccccc2)c2n1CCC2

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGES O14684 2/20 0.44
ALOX5 P09917 15/20 0.44
PTGS1 P23219 2/20 0.43
DHFR P00374 1/20 0.35
PTGS2 P35354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458748 0.84 ALOX5 (0.46) PTGESALOX5PTGS1DHFR
SCHEMBL9459144 0.78 PTGES (0.53) PTGESALOX5PTGS1
SCHEMBL9458881 0.76 OXER1 (0.52) PTGESALOX5PTGS1
SCHEMBL9458593 0.75 ALOX5 (0.65) PTGESALOX5PTGS1
SCHEMBL9458745 0.75 ALOX5 (0.65) PTGESALOX5PTGS1
SCHEMBL8594214 0.69 PTGES (0.74) PTGESALOX5PTGS1
SCHEMBL9458661 0.69 CYP2D6 (0.39) PTGS1PTGS2
SCHEMBL1785116 0.69 PTGES (0.38) PTGESDHFR
SCHEMBL9472243 0.68 PTGS2 (0.49) ALOX5PTGS1DHFRPTGS2
SCHEMBL10445152 0.68 CYP2D6 (0.37) ALOX5PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260451-A Enzyme inhibitors MERCKLE GMBH (DE) 1993-11-09 US disclosed
EP-0397175-A1 Substituted pyrrolizine compounds and theit use as pharmaceuticals Dannhardt, Gerd, Prof.Dr. (DE) 1990-11-14 EP disclosed