SCHEMBL9458661

SCHEMBL9458661

CCCCCCc1cc(-c2ccccc2)c2n1CCC2

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.39
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
HSD11B1 P28845 1/20 0.35
SOAT1 P35610 3/20 0.35
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10445152 0.99 CYP2D6 (0.37) CYP2D6CNR1CNR2HRH3HSD11B1
SCHEMBL6475630 0.74 ALOX5 (0.45) PTGS1
SCHEMBL9537195 0.72 PTGS2 (0.49) HRH3HSD11B1PTGS1PTGS2
SCHEMBL9458748 0.69 ALOX5 (0.46) PTGS1
SCHEMBL9458649 0.69 PTGES (0.44) PTGS1PTGS2
SCHEMBL9472243 0.67 PTGS2 (0.49) HRH3PTGS1PTGS2
SCHEMBL5672731 0.65 SOAT1 (0.54) SOAT1
SCHEMBL25867877 0.64 LIPG (0.47) HSD11B1SOAT1
SCHEMBL8521601 0.64 LIPG (0.55) SOAT1
SCHEMBL3726514 0.64 LIPG (0.55) SOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260451-A Enzyme inhibitors MERCKLE GMBH (DE) 1993-11-09 US disclosed
EP-0397175-A1 Substituted pyrrolizine compounds and theit use as pharmaceuticals Dannhardt, Gerd, Prof.Dr. (DE) 1990-11-14 EP disclosed