SCHEMBL9463517

SCHEMBL9463517

CCSCCC(C(C)=O)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.43
BHMT Q93088 4/20 0.38
NOS2 P35228 2/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
METAP2 P50579 4/20 0.36
BHMT2 Q9H2M3 1/20 0.36
METAP1 P53582 2/20 0.36
CHRM1 P11229 1/20 0.34
AKR1A1 P14550 1/20 0.34
CHRM3 P20309 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
ADRA1A P35348 1/20 0.34
HRH1 P35367 1/20 0.34
DRD3 P35462 1/20 0.34
SLC6A3 Q01959 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4953418 0.89 TSHR (0.48) TSHRBHMTNOS2NOS3NOS1
SCHEMBL15948621 0.80 METAP2 (0.46) TSHRMETAP2METAP1TDP1
SCHEMBL16123404 0.77 METAP2 (0.38) TSHRMETAP2METAP1
SCHEMBL721101 0.77 GPR84 (0.50) TSHRBHMTMETAP2BHMT2METAP1
SCHEMBL9463332 0.77 RNPEP (0.56) RNPEP
SCHEMBL9392724 0.75 CHRM1 (0.41) CHRM1AKR1A1CHRM3HTR2AHTR2C
Ethionine SCHEMBL15005828 0.75 BHMT (0.59) BHMTNOS2NOS3NOS1BHMT2
Ethionine SCHEMBL31087565 0.75 BHMT (0.59) BHMTNOS2NOS3NOS1BHMT2
Ethionine SCHEMBL8967 0.74 BHMT (0.63) BHMTNOS2NOS3NOS1BHMT2
Ethionine SCHEMBL8966 0.74 BHMT (0.63) BHMTNOS2NOS3NOS1BHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5177211-A Anti-platelet aggregation and anti-hypotensive ALTER, S.A. (ES) 1993-01-05 US disclosed
EP-0325187-B1 4-ALKYL-1, 4-DIHYDROPYRIDINES WITH PAF-ANTAGONIST ACTIVITY ALTER, S.A. (ES) 1992-11-11 EP disclosed
EP-0325187-A1 4-alkyl-1, 4-dihydropyridines with PAF-antagonist activity ALTER, S.A. (ES) 1989-07-26 EP disclosed