SCHEMBL9464640

SCHEMBL9464640

O=S(=O)(Nc1ccc(I)cc1F)c1cccc2ccccc12

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.62
SLC16A3 O15427 3/20 0.49
PGAM1 P18669 2/20 0.47
HCRTR1 O43613 1/20 0.47
TSHR P16473 1/20 0.45
PGR P06401 1/20 0.45
RORA P35398 1/20 0.44
RORC P51449 1/20 0.44
NR1H2 P55055 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
MCL1 Q07820 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43
PFKFB3 Q16875 1/20 0.43
TYMS P04818 1/20 0.43
EDNRB P24530 1/20 0.42
EDNRA P25101 1/20 0.42
RECQL P46063 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29559690 0.82 ACLY (0.43) ACLYSLC16A3PGRMCL1PKM
SCHEMBL21545890 0.82 ACLY (0.43) ACLYSLC16A3PGRMCL1PKM
SCHEMBL9465779 0.80 MEN1 (0.58) TSHRALDH1A1
SCHEMBL2146366 0.78 PTGES2 (0.61) ACLY
SCHEMBL9616624 0.77 ALDH1A1 (0.56) HCRTR1TSHRPGRRORARORC
SCHEMBL9464328 0.77 MAP2K1 (0.61) ACLYTSHRALDH1A1HTT
SCHEMBL21999593 0.76 ACLY (1.00) ACLY
SCHEMBL9464387 0.74 SLC40A1 (0.51) ACLYTSHR
SCHEMBL6717132 0.73 ACLY (0.54) ACLYTSHRHTT
SCHEMBL2146100 0.73 MCL1 (0.51) ACLYTSHRMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258399-A 5-lipoxygenase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-11-02 US disclosed
US-5236948-A Lipoxygenase inhibitor IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-08-17 US disclosed
EP-0495594-A1 Sulphonamide derivatives ZENECA LIMITED (GB) 1992-07-22 EP disclosed