SCHEMBL9466971

SCHEMBL9466971

CCCCC(C(=O)OCC)C(C)(O)c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 3/20 0.46
KCNH2 Q12809 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.44
LMNA P02545 3/20 0.42
TDP1 Q9NUW8 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
TBXAS1 P24557 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TSHR P16473 2/20 0.38
RORC P51449 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
PKM P14618 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9720312 0.86 TBXAS1 (0.50) KCNA5KCNH2L3MBTL1LMNATDP1
Ammonia Solution, Strong SCHEMBL9720296 0.85 TBXAS1 (0.49) KCNA5KCNH2L3MBTL1LMNATDP1
SCHEMBL9720329 0.85 KCNA5 (0.47) KCNA5KCNH2L3MBTL1LMNATDP1
SCHEMBL10904085 0.84 TDP1 (0.44) TDP1CYP3A4SMN1; SMN2TSHRKMT2A
SCHEMBL11075778 0.79 ALOX5 (0.38) L3MBTL1LMNATDP1CYP1A2MAPK1
SCHEMBL9466966 0.78 CYP3A4 (0.41) KCNA5LMNATDP1CYP1A2CYP3A4
Piperidine SCHEMBL9720307 0.77 KCNA5 (0.43) KCNA5KCNH2L3MBTL1LMNATDP1
SCHEMBL10904098 0.76 POLB (0.49) TDP1SMN1; SMN2TSHRCYP2C19KMT2A
SCHEMBL11067677 0.73 TDP1 (0.35) L3MBTL1LMNATDP1CYP3A4TSHR
Iodide SCHEMBL9340453 0.73 L3MBTL1 (0.47) L3MBTL1LMNACYP1A2TBXAS1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4479003-A Heterocyclic-hydroxy-substituted carboxylate esters PHILIP MORRIS, INCORPORATED (US) 1984-10-23 US claimed
EP-0037163-A2 Flavouring agents, smoking compositions, combustible articles and foodstuffs containing such agents, and a method of producing the same PHILIP MORRIS INCORPORATED (US) 1981-10-07 EP claimed
US-5256785-A Smoking compositions containing an oxalate flavorant-release additive PHILIP MORRIS INCORPORATED (US) 1993-10-26 US disclosed
US-5218118-A Smoking compositions containing a pyrazine-ethanol flavorant-release additive PHILIP MORRIS INCORPORATED (US) 1993-06-08 US disclosed
US-5174308-A SMOKING COMPOSITIONS CONTAINING A PYRAZINEETHANOL FLAVORANT-RELEASE ADDITIVE PHILIP MORRIS INCORPORATED (US) 1992-12-29 US disclosed
US-5172706-A Smoking compositions containing an oxalate flavorant-release additive PHILIP MORRIS INCORPORATED (US) 1992-12-22 US disclosed
EP-0518617-A1 Smoking compositions containing a pyrazineethanol flavorant-release additive Philip Morris Products Inc. (US) 1992-12-16 EP disclosed
US-5080719-A Pyrazine derivatives PHILIP MORRIS INCORPORATED (US) 1992-01-14 US disclosed
US-4872918-A Heterocyclic esters and smoking compositions containing a heterocyclic ester flavorant-release additive PHILIP MORRIS INCORPORATED (US) 1989-10-10 US disclosed
EP-0309203-A2 Flavorant-release additives and compositions containing them Philip Morris Products Inc. (US) 1989-03-29 EP disclosed
US-4701282-A CIGARETTES PHILIP MORRIS INCORPORATED (US) 1987-10-20 US disclosed
US-4690157-A DERIVATIVES OF BUTYROLACTONE OR VALEROLACTONE; CIGARETTES PHILIP MORRIS INCORPORATED (US) 1987-09-01 US disclosed
US-4538627-A Smoking compositions containing a β-hydroxy-γ-ketoester flavorant-release additive PHILIP MORRIS INCORPORATED (US) 1985-09-03 US disclosed
US-4479003-A Heterocyclic-hydroxy-substituted carboxylate esters PHILIP MORRIS, INCORPORATED (US) 1984-10-23 US disclosed
US-4479003-A Heterocyclic-hydroxy-substituted carboxylate esters PHILIP MORRIS, INCORPORATED (US) 1984-10-23 US disclosed
US-4312368-A Smoking compositions PHILIP MORRIS, INCORPORATED (US) 1982-01-26 US disclosed
US-4312368-A Smoking compositions PHILIP MORRIS, INCORPORATED (US) 1982-01-26 US disclosed
EP-0037163-A2 Flavouring agents, smoking compositions, combustible articles and foodstuffs containing such agents, and a method of producing the same PHILIP MORRIS INCORPORATED (US) 1981-10-07 EP disclosed