SCHEMBL9467343

SCHEMBL9467343

c1ccc(CC2COC(N3CCN(CCCC4CCc5ccccc54)CC3)CO2)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.51
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
ABCB1 P08183 1/20 0.41
CHRM5 P08912 1/20 0.41
ADRA2A P08913 1/20 0.41
CHRM1 P11229 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
CHRM3 P20309 1/20 0.41
KCNH2 Q12809 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
HTR1A P08908 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1038534 0.94 SIGMAR1 (0.43) SIGMAR1
SCHEMBL9466307 0.88 SIGMAR1 (0.51) SIGMAR1
SCHEMBL9174172 0.88 SIGMAR1 (0.43) SIGMAR1ADRA2AADRA2BADRA2CHTR1A
SCHEMBL9175467 0.83 SIGMAR1 (0.40) SIGMAR1KCNH2TMEM97HTR1A
SCHEMBL9467124 0.82 ALDH1A1 (0.36)
SCHEMBL9175775 0.80 SIGMAR1 (0.45) SIGMAR1CHRM2CHRM4ABCB1CHRM5
SCHEMBL8303444 0.80 SIGMAR1 (0.55) SIGMAR1
SCHEMBL9181626 0.80 PTGDR2 (0.39)
SCHEMBL9178363 0.78 SIGMAR1 (0.41) SIGMAR1HTR1A
SCHEMBL9178801 0.75 CRBN (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5194437-A Substituted with oxygen containing heterocycle, central nervous system disorders, neuroendocrine disorders ADIR ET COMPAGNIE (FR) 1993-03-16 US disclosed