SCHEMBL9470265

SCHEMBL9470265

O=CONC1N=C(c2ccccc2)c2ccccc2-n2cnnc21

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 10/20 0.60
BRD4 O60885 8/20 0.40
BRD2 P25440 8/20 0.40
BRD3 Q15059 8/20 0.40
CCKAR P32238 2/20 0.39
SENP1 Q9P0U3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9470619 0.79 BRD4 (0.64) CCKBRBRD4BRD2BRD3
Formic Acid SCHEMBL9470262 0.77 CCKBR (0.53) CCKBRBRD4BRD2BRD3CCKAR
SCHEMBL9469852 0.75 CCKBR (1.00) CCKBRBRD4BRD2BRD3SENP1
SCHEMBL9470437 0.72 CCKBR (1.00) CCKBR
SCHEMBL9645886 0.70 CCKBR (0.73) CCKBRCCKAR
SCHEMBL9648025 0.67 CCKBR (0.75) CCKBRBRD4BRD2BRD3CCKAR
SCHEMBL11034765 0.67 OPRK1 (0.55) CCKBRBRD4BRD2BRD3
SCHEMBL11734724 0.66 CCKBR (0.56) CCKBRBRD4BRD2BRD3CCKAR
SCHEMBL9469193 0.65 CCKBR (1.00) CCKBRBRD4BRD2BRD3SENP1
SCHEMBL11638117 0.62 CCKBR (0.45) CCKBRBRD4BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5185331-A Administering to treat panic and anxiety disorders MERCK & CO., INC. (US) 1993-02-09 US disclosed
EP-0514125-A1 Triazolobenzodiazepines MERCK & CO. INC. (US) 1992-11-19 EP disclosed