SCHEMBL9470868

SCHEMBL9470868

CS(=O)(=O)Nc1ccc(OCC(O)CN2CCC(C(=O)c3ccc(NS(C)(=O)=O)cc3)CC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.65
ADRB1 P08588 7/20 0.65
ADRB3 P13945 7/20 0.65
KCNH2 Q12809 3/20 0.61
SMN1; SMN2 Q16637 1/20 0.55
MAPT P10636 2/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
ABCB1 P08183 2/20 0.51
KDM4E B2RXH2 1/20 0.51
POLB P06746 1/20 0.51
SCN1A P35498 1/20 0.49
SCN5A Q14524 1/20 0.49
SCN9A Q15858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9471731 0.83 LTA4H (0.63) KCNH2CYP3A4CYP2D6CYP2C19KDM4E
SCHEMBL9444448 0.82 KCNH2 (0.56) ADRB2ADRB1ADRB3KCNH2SMN1; SMN2
SCHEMBL10580036 0.82 KCNH2 (0.56) ADRB2ADRB1ADRB3KCNH2SMN1; SMN2
SCHEMBL9444381 0.79 KCNH2 (0.56) ADRB2ADRB1ADRB3KCNH2SMN1; SMN2
SCHEMBL12722227 0.79 CYP2D6 (0.69) ADRB2ADRB1ADRB3SMN1; SMN2MAPT
SCHEMBL9444349 0.79 KCNH2 (0.62) KCNH2SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL9839933 0.79 ADRB2 (1.00) ADRB2ADRB1ADRB3KCNH2MAPT
SCHEMBL9480753 0.79 LTA4H (0.57) KCNH2CYP3A4CYP2D6CYP2C19KDM4E
Hydrochloric Acid SCHEMBL9444401 0.78 KCNH2 (0.62) KCNH2SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL12722228 0.77 CACNA1G (0.64) ADRB2ADRB1ADRB3KCNH2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5202346-A Antiarrhythmic agent AMERICAN HOME PRODUCTS CORPORATION (US) 1993-04-13 US claimed
US-5254689-A Antiarrhythmia agents AMERICAN HOME PRODUCTS CORPORATION (US) 1993-10-19 US disclosed