SCHEMBL9475563

SCHEMBL9475563

CC1(C)N=C(c2cccc[n+]2[O-])c2cc(Cl)ccc2O1

nearest known ligand 0.31

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.31
ABCC9 O60706 2/20 0.31
ABCC8 Q09428 2/20 0.31
KCNJ11 Q14654 2/20 0.31
KCNJ8 Q15842 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MAPK1 P28482 1/20 0.31
KCNK2 O95069 1/20 0.31
ADRB2 P07550 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
HTR1A P08908 1/20 0.31
CHRM5 P08912 1/20 0.31
ADRA2A P08913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9476674 0.86 ABCC9 (0.32) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9475319 0.85 ABCC9 (0.31) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9476803 0.82 ABCC9 (0.32) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8027470 0.82
SCHEMBL9476372 0.82 L3MBTL1 (0.36) CHRM1ALDH1A1LMNACHRM2HTR1A
SCHEMBL9475710 0.82 ABCC9 (0.41) CHRM1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9475265 0.82 ABCC9 (0.50) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9478300 0.82 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9476029 0.81 ABCC9 (0.32) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9475663 0.81 ALOX5 (0.34) ABCC9ABCC8KCNJ11KCNJ8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0477789-A1 1,3-Benzoxazine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1992-04-01 EP claimed
US-5270308-A Hypotensives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-12-14 US disclosed
CN-1060467-A 1,3-benzoxazine derivatives, its production method and purposes TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1992-04-22 CN disclosed
EP-0477789-A1 1,3-Benzoxazine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1992-04-01 EP disclosed