SCHEMBL9478024

SCHEMBL9478024

CCN(CC)CC(O)CSC(C#N)=C1NCCc2cc(OC)c(OC)cc21

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
CHEK1 O14757 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
HSP90AB1 P08238 1/20 0.30
S1PR2 O95136 1/20 0.30
HPGD P15428 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9476039 0.99 KMT2A (0.33) KMT2AMEN1CHEK1CYP1A2CYP3A4
SCHEMBL9475901 0.91 ACHE (0.38) MAPK1
SCHEMBL9477129 0.91 KMT2A (0.32) KMT2AMEN1CHEK1
Hydrochloric Acid SCHEMBL9476844 0.91 ACHE (0.37) MAPK1
Hydrochloric Acid SCHEMBL9479486 0.90 KMT2A (0.32) KMT2AMEN1CHEK1
SCHEMBL9477694 0.83 ABCC4 (0.36)
SCHEMBL9476703 0.83 KMT2A (0.33) KMT2AMEN1CYP2D6HSD17B10
Hydrochloric Acid SCHEMBL9478051 0.83 ABCC4 (0.36)
SCHEMBL9475100 0.82 KMT2A (0.33) KMT2AMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL9475282 0.82 KDM4E (0.35) KMT2AMEN1HSD17B10S1PR2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5179089-A Antiallergens, asthma CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1993-01-12 US claimed
EP-0486211-A1 Isoquinoline derivatives CHINOIN Gyògyszer és Vegyészeti Termékek Gyára RT. (HU) 1992-05-20 EP claimed
JP-4283567-A None JP disclosed
JP-H04283567-A NEW COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING NEW COMPOUND AND ITS PRODUCTION CHINOIN GYOGYSZER V T G RT 1992-10-08 JP disclosed