SCHEMBL9475901

SCHEMBL9475901

CCOc1cc2c(cc1OCC)C(=C(C#N)SCC(O)CN(CC)CC)NCC2

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.38
ABCC4 O15439 1/20 0.38
ABCB11 O95342 1/20 0.38
CHRM2 P08172 1/20 0.38
ADRA2A P08913 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CHRM1 P11229 1/20 0.38
PTGS1 P23219 1/20 0.38
PDE4A P27815 1/20 0.38
SLC6A4 P31645 1/20 0.38
KCNH2 Q12809 1/20 0.38
MAPK1 P28482 1/20 0.31
CASP1 P29466 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9476844 0.99 ACHE (0.37) ACHEABCC4ABCB11CHRM2ADRA2A
SCHEMBL9477694 0.92 ABCC4 (0.36) ACHEABCC4ABCB11CHRM2ADRA2A
SCHEMBL9478024 0.91 KMT2A (0.33) MAPK1
Hydrochloric Acid SCHEMBL9478051 0.91 ABCC4 (0.36) ACHEABCC4ABCB11CHRM2ADRA2A
Hydrochloric Acid SCHEMBL9476039 0.91 KMT2A (0.33)
SCHEMBL9479120 0.84 ABCC4 (0.37) ACHEABCC4ABCB11CHRM2ADRA2A
SCHEMBL9476362 0.83 ADRA2A (0.37) ACHEABCC4ABCB11CHRM2ADRA2A
SCHEMBL9476649 0.83 ABCC4 (0.37) ACHEABCC4ABCB11CHRM2ADRA2A
Hydrochloric Acid SCHEMBL9477019 0.83 ABCC4 (0.37) ACHEABCC4ABCB11CHRM2ADRA2A
SCHEMBL9476660 0.83 ABCC4 (0.36) ACHEABCC4ABCB11CHRM2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5179089-A Antiallergens, asthma CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1993-01-12 US claimed
EP-0486211-A1 Isoquinoline derivatives CHINOIN Gyògyszer és Vegyészeti Termékek Gyára RT. (HU) 1992-05-20 EP claimed