SCHEMBL9477694

SCHEMBL9477694

CCOc1cc2c(cc1OCC)C(=C(C#N)SCC(O)CN(CCO)CCO)NCC2

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCC4 O15439 1/20 0.36
ABCB11 O95342 1/20 0.36
CHRM2 P08172 1/20 0.36
ADRA2A P08913 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
CHRM1 P11229 1/20 0.36
ACHE P22303 1/20 0.36
PTGS1 P23219 1/20 0.36
PDE4A P27815 1/20 0.36
SLC6A4 P31645 1/20 0.36
KCNH2 Q12809 1/20 0.36
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9478051 0.99 ABCC4 (0.36) ABCC4ABCB11CHRM2ADRA2AADORA3
SCHEMBL9475901 0.92 ACHE (0.38) ABCC4ABCB11CHRM2ADRA2AADORA3
SCHEMBL9477129 0.91 KMT2A (0.32) PDE4A
Hydrochloric Acid SCHEMBL9476844 0.91 ACHE (0.37) ABCC4ABCB11CHRM2ADRA2AADORA3
Hydrochloric Acid SCHEMBL9479486 0.90 KMT2A (0.32) PDE4A
SCHEMBL9478024 0.83 KMT2A (0.33)
Hydrochloric Acid SCHEMBL9476039 0.83 KMT2A (0.33)
SCHEMBL9479120 0.82 ABCC4 (0.37) ABCC4ABCB11CHRM2ADRA2AADORA3
SCHEMBL9476362 0.81 ADRA2A (0.37) ABCC4ABCB11CHRM2ADRA2AADORA3
SCHEMBL9476649 0.81 ABCC4 (0.37) ABCC4ABCB11CHRM2ADRA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5179089-A Antiallergens, asthma CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1993-01-12 US claimed
EP-0486211-A1 Isoquinoline derivatives CHINOIN Gyògyszer és Vegyészeti Termékek Gyára RT. (HU) 1992-05-20 EP claimed