SCHEMBL9478784

SCHEMBL9478784

O=C(Nc1ccc(C(F)(F)F)cc1)NS(=O)(=O)c1ccc2c(c1)C=CC2

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.49
CA1 P00915 5/20 0.49
CA2 P00918 5/20 0.49
CA9 Q16790 5/20 0.49
MAPT P10636 2/20 0.49
HRH3 Q9Y5N1 5/20 0.48
KCNH2 Q12809 1/20 0.47
EPHX2 P34913 4/20 0.46
KCNA1 Q09470 1/20 0.43
KCNAB1 Q14722 1/20 0.43
IDH1 O75874 1/20 0.43
IDO1 P14902 1/20 0.42
TP53 P04637 2/20 0.42
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9478543 0.91 HRH3 (0.49) CA12CA1CA2CA9MAPT
SCHEMBL9478237 0.87 TP53 (0.56) CA12CA1CA2CA9KCNA1
SCHEMBL9478847 0.86 MEN1 (0.47) CA1CA2CA9EPHX2KCNA1
SCHEMBL9478381 0.85 CA1 (0.46) CA12CA1CA2CA9KCNA1
SCHEMBL7983217 0.85 KCNA1 (0.53) CA12CA1CA2CA9MAPT
SCHEMBL9479492 0.84 CA1 (0.40) CA12CA1CA2CA9MAPT
SCHEMBL9478768 0.84 CA2 (0.44) CA1CA2CA9MAPTKCNA1
SCHEMBL9477487 0.83 MEN1 (0.60) CA12CA2CA9MAPTKCNA1
SCHEMBL9477595 0.81 EPHX1 (0.47) CA12CA1CA2CA9MAPT
SCHEMBL9478165 0.81 MEN1 (0.48) CA12CA1CA2CA9KCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5262440-A Treatment of neoplasms ELI LILLY AND COMPANY (US) 1993-11-16 US disclosed
EP-0546763-A1 Antitumor compositions and methods of treatment ELI LILLY AND COMPANY (US) 1993-06-16 EP disclosed