SCHEMBL9482240

SCHEMBL9482240

CS(=O)(=O)Nc1cccc2coc(C(=O)NC3CCN(Cc4ccccc4)CC3)c12

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.53
SIGMAR1 Q99720 5/20 0.52
SLC6A12 P48065 2/20 0.51
SLC6A13 Q9NSD5 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
POLB P06746 1/20 0.50
RAB9A P51151 1/20 0.50
MAOB P27338 1/20 0.48
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
TMEM97 Q5BJF2 2/20 0.48
MCHR1 Q99705 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9481804 0.93 MCHR1 (0.47) DRD4SIGMAR1SLC6A12SLC6A13RAB9A
SCHEMBL9482200 0.86 DRD4 (0.38) DRD4SIGMAR1SLC6A12SLC6A13L3MBTL1
SCHEMBL9483648 0.81 DRD4 (0.52) DRD4SLC6A12SLC6A13MAOBKMT2A
SCHEMBL9482226 0.80 SIGMAR1 (0.55) DRD4SIGMAR1SLC6A12SLC6A13L3MBTL1
SCHEMBL9852247 0.80 SIGMAR1 (0.59) DRD4SIGMAR1SLC6A12SLC6A13L3MBTL1
SCHEMBL9727135 0.80 DRD4 (0.67) DRD4SIGMAR1SLC6A12SLC6A13L3MBTL1
Dimethylamine SCHEMBL9852061 0.79 DRD4 (0.63) DRD4SIGMAR1SLC6A12SLC6A13POLB
SCHEMBL9727088 0.76 DRD4 (0.62) DRD4SIGMAR1SLC6A12MAOBMCHR1
SCHEMBL9727190 0.76 DRD4 (0.62) DRD4SIGMAR1MAOBMCHR1
SCHEMBL9727173 0.73 SIGMAR1 (0.57) DRD4SIGMAR1SLC6A12SLC6A13MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210090-A Antiarrythmia G. D. SEARLE & CO. (US) 1993-05-11 US claimed
EP-0416581-A1 Substituted N-benzylpiperidine amides G.D. Searle & Co. (US) 1991-03-13 EP claimed
US-5210090-A Antiarrythmia G. D. SEARLE & CO. (US) 1993-05-11 US disclosed
EP-0416581-A1 Substituted N-benzylpiperidine amides G.D. Searle & Co. (US) 1991-03-13 EP disclosed