SCHEMBL9495668

SCHEMBL9495668

COc1cccc2c1CC(OCc1ccccc1)C2=O

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.55
CYP19A1 P11511 2/20 0.50
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
DRD2 P14416 1/20 0.41
NAAA Q02083 1/20 0.40
HTT P42858 1/20 0.40
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HTR1A P08908 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3602309 0.77 ACHE (0.46) ACHECYP19A1KDM4EMAPT
SCHEMBL9495652 0.73 MEN1 (0.45) ACHEMAPTHTTNPC1RAB9A
SCHEMBL14939214 0.73 ACHE (0.62) ACHECYP19A1KDM4ELMNAPOLB
SCHEMBL27532854 0.71 ALDH1A1 (0.52) ACHECYP19A1KDM4EMAPTDRD2
SCHEMBL15746282 0.71 ACHE (1.00) ACHECYP19A1KDM4ELMNAPOLB
SCHEMBL31297867 0.71 ACHE (0.70) ACHECYP19A1KDM4ELMNAPOLB
SCHEMBL11204280 0.70 HTT (0.51) LMNAPOLBMAPTHTT
SCHEMBL25604493 0.70 ACHE (0.68) ACHECYP19A1CA1CA2KDM4E
SCHEMBL30070593 0.70 PSEN1 (0.33) ACHECA1CA2
SCHEMBL28529968 0.70 ACHE (0.62) ACHECYP19A1CA1CA2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0522000-A1 5-LIPOXYGENASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1993-01-13 EP disclosed
WO-1991014674-A2 5-LIPOXYGENASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1991-10-03 WO disclosed