SCHEMBL9501142

SCHEMBL9501142

CC(C)COC(=O)C(N)C1CN=C(c2ccccc2F)c2ccccc2N1C

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 6/20 0.47
OPRD1 P41143 4/20 0.46
OPRK1 P41145 4/20 0.46
OPRM1 P35372 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11142686 0.80 CCKBR (0.47) CCKBROPRD1OPRK1OPRM1
SCHEMBL9501135 0.79 CCKBR (0.64) CCKBROPRD1OPRK1OPRM1
SCHEMBL11138052 0.78 CCKBR (0.45) CCKBROPRD1OPRK1OPRM1
SCHEMBL11144864 0.78 OPRK1 (0.47) CCKBROPRD1OPRK1OPRM1
SCHEMBL10863771 0.77 CCKBR (0.63) CCKBROPRD1OPRK1OPRM1
SCHEMBL10865137 0.77 OPRD1 (0.62) CCKBROPRD1OPRK1OPRM1
SCHEMBL11006750 0.76 CCKBR (0.49) CCKBROPRD1OPRK1OPRM1
Hydrochloric Acid SCHEMBL11167236 0.76 OPRD1 (0.61) CCKBROPRD1OPRK1OPRM1
SCHEMBL9531702 0.73 CCKBR (0.67) CCKBROPRD1OPRK1OPRM1
SCHEMBL9499795 0.73 CCKBR (0.58) CCKBROPRD1OPRK1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5206238-A Cholecystokinin antagonists MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0486271-A2 Cholecystokinin antagonists for treating neurological disorders MERCK & CO. INC. (US) 1992-05-20 EP disclosed