SCHEMBL9501587

SCHEMBL9501587

Nc1ccc2c(c1)C(=O)N(CCO)CCO2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
SCN1A P35498 1/20 0.38
SCN4A P35499 1/20 0.38
KCNH2 Q12809 1/20 0.38
SCN5A Q14524 1/20 0.38
SCN9A Q15858 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
SCN8A Q9UQD0 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
ROCK2 O75116 1/20 0.37
PRMT5 O14744 11/20 0.36
WDR77 Q9BQA1 11/20 0.36
ALPL P05186 1/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 1/20 0.36
CASP1 P29466 2/20 0.35
HSD17B10 Q99714 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8640110 0.86 ALDH1A1 (0.40) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL24170261 0.83 NOS3 (0.41) KDM4EALDH1A1HPGDSCN1ASCN4A
SCHEMBL15264451 0.80 NOS3 (0.39) KDM4EALDH1A1KCNH2GAAMAPT
SCHEMBL9504216 0.80 PIK3CD (0.43) ALDH1A1MAPTCASP1MEN1KMT2A
SCHEMBL9501566 0.79 RAF1 (0.40) KDM4EALDH1A1GAAMAPTCASP1
SCHEMBL29631754 0.77 NOS3 (0.40) KDM4EKCNH2GAAMAPTKMT2A
SCHEMBL11969208 0.77 NOS3 (0.40) KDM4EKCNH2GAAMAPTKMT2A
SCHEMBL19138468 0.76 ALPL (0.49) KDM4ESCN1ASCN4AKCNH2SCN5A
SCHEMBL14480886 0.74 KCNH2 (0.69) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL8641707 0.72 ALDH1A1 (0.37) KDM4EALDH1A1HPGDGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0355598-B1 BETA-PHENOXYETHYL AMINES AND THEIR USE IN THE PREPARATION OF DYES BAYER AG (DE) 1993-06-16 EP disclosed
US-5126481-A Cyclization, reduction, decyclization BAYER AKTIENGESELLSCHAFT (DE) 1992-06-30 US disclosed
US-5041629-A Beta-phenoxyethylamines and their use for the preparation of dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1991-08-20 US disclosed
EP-0355598-A2 Beta-phenoxyethyl amines and their use in the preparation of dyes BAYER AG (DE) 1990-02-28 EP disclosed