SCHEMBL9501566

SCHEMBL9501566

CN1CCOc2ccc(N)cc2C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 1/20 0.40
GAA P10253 2/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
PKM P14618 2/20 0.38
LRRK2 Q5S007 1/20 0.38
ALDH1A1 P00352 2/20 0.36
CASP1 P29466 2/20 0.36
CASP7 P55210 2/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
AR P10275 1/20 0.36
NOTUM Q6P988 1/20 0.36
LMNA P02545 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2060409 0.88 GAA (0.40) RAF1GAAMAPTKDM4ELRRK2
SCHEMBL10274465 0.83 PIK3CA (0.52) GAAMAPTKDM4EPKMALDH1A1
SCHEMBL9501587 0.79 KDM4E (0.38) GAAMAPTKDM4EALDH1A1CASP1
SCHEMBL24170261 0.78 NOS3 (0.41) KDM4EALDH1A1
SCHEMBL30781179 0.78 GAA (0.46) GAAMAPTKDM4EPKMALDH1A1
SCHEMBL519949 0.78 GAA (0.46) GAAMAPTKDM4EPKMALDH1A1
SCHEMBL31707229 0.77 PKM (0.44) PKMNPC1TSHRARNOTUM
SCHEMBL16546168 0.77 PKM (0.44) PKMNPC1TSHRARNOTUM
SCHEMBL9501575 0.77 PIK3CD (0.49) MAPTALDH1A1CASP1CASP7NPC1
SCHEMBL14995200 0.76 HTR3A (0.47) GAALRRK2ARMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0355598-B1 BETA-PHENOXYETHYL AMINES AND THEIR USE IN THE PREPARATION OF DYES BAYER AG (DE) 1993-06-16 EP disclosed
US-5126481-A Cyclization, reduction, decyclization BAYER AKTIENGESELLSCHAFT (DE) 1992-06-30 US disclosed
US-5041629-A Beta-phenoxyethylamines and their use for the preparation of dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1991-08-20 US disclosed
EP-0355598-A2 Beta-phenoxyethyl amines and their use in the preparation of dyes BAYER AG (DE) 1990-02-28 EP disclosed