SCHEMBL9501704

SCHEMBL9501704

O=C([C@@H]1CCCN1C(=O)CCCc1cccc(Oc2ccccc2)c1)N1CCCC1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PREP P48147 3/20 0.53
FFAR1 O14842 1/20 0.50
HTR1A P08908 1/20 0.49
HTR2A P28223 1/20 0.49
HTR7 P34969 1/20 0.49
HTR6 P50406 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9500400 0.89 ACE (0.52)
SCHEMBL6285952 0.88 PREP (0.65) PREP
SCHEMBL6285958 0.88 PREP (0.65) PREP
SCHEMBL10339417 0.86 PREP (0.65) PREP
SCHEMBL9501238 0.86 FKBP1A (0.54) FFAR1
SCHEMBL31324093 0.78 DPP4 (0.58) HTR1AHTR7
SCHEMBL9501712 0.77 PREP (0.48) PREP
SCHEMBL8153242 0.76 MEN1 (0.55) PREP
SCHEMBL8153245 0.76 MEN1 (0.55) PREP
SCHEMBL7330019 0.76 MEN1 (0.63)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0232849-B1 PYRROLIDINEAMIDE DERIVATIVE OF ACYLAMINO ACID, PHARMACEUTICAL COMPOSITION AND USE SUNTORY LIMITED (JP) 1993-05-05 EP disclosed
US-5198458-A Pyrrolidineamide derivatives of acylamino acid and pharmaceutical composition containing the same SUNTORY LIMITED (JP) 1993-03-30 US disclosed
US-4826870-A CURING AMNESIA SUNTORY LIMITED (JP) 1989-05-02 US disclosed
EP-0232849-A2 Pyrrolidineamide derivative of acylamino acid, pharmaceutical composition and use SUNTORY LIMITED (JP) 1987-08-19 EP disclosed