SCHEMBL9502783

SCHEMBL9502783

COc1ccc2c(ccn2CCCCc2ccccn2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.48
ITGAV P06756 3/20 0.48
ITGB5 P18084 2/20 0.48
HRH1 P35367 1/20 0.46
HTR6 P50406 1/20 0.46
HTR2C P28335 2/20 0.45
MTNR1A P48039 1/20 0.45
MTNR1B P49286 1/20 0.45
KDM4E B2RXH2 1/20 0.44
GLA P06280 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMPD1 P17405 1/20 0.43
ITGB1 P05556 1/20 0.42
ITGA5 P08648 1/20 0.42
CDK4 P11802 2/20 0.42
CCND1 P24385 2/20 0.42
PLA2G2A P14555 1/20 0.42
KCNA5 P22460 1/20 0.42
CYP24A1 Q07973 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14300254 0.86 ITGB3 (0.45) ITGB3ITGAVITGB5ITGB1ITGA5
SCHEMBL8845546 0.84 ITGB3 (0.48) ITGB3ITGAVITGB5MTNR1AMTNR1B
SCHEMBL8845779 0.83 CDK4 (0.44) ITGB3ITGAVITGB5HRH1CDK4
SCHEMBL14274529 0.83 MCL1 (0.44) ITGB3ITGAVITGB5NPC1RAB9A
SCHEMBL9502777 0.79 SLC6A2 (0.48) HRH1HTR6HTR2CMTNR1AMTNR1B
SCHEMBL8845730 0.79 ITGB3 (0.47) ITGB3ITGAVITGB5ITGB1ITGA5
SCHEMBL8845545 0.78 ITGB3 (0.44) ITGB3ITGAVITGB5ITGB1ITGA5
SCHEMBL18856948 0.76 MTNR1A (0.58) HTR2CMTNR1AMTNR1BKDM4ECDK4
SCHEMBL4394621 0.75 MTNR1A (0.56) HTR2CMTNR1AMTNR1BKDM4ECDK4
SCHEMBL5841872 0.75 HTR2C (0.55) HTR2CMTNR1AMTNR1BKDM4ECDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5214058-A Acetylcholinesterase inhibitors, treatment of senile dementia HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-05-25 US claimed
US-5214058-A Acetylcholinesterase inhibitors, treatment of senile dementia HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-05-25 US disclosed
EP-0471296-A1 1-(Pyridinylalkyl)-1H-indoles, indolines and related analogs HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-02-19 EP disclosed