SCHEMBL9503471

SCHEMBL9503471

COC(=O)c1cc(C(O)CNCC2CCc3ccccc3C2=O)ccc1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 11/20 0.55
ADRB1 P08588 9/20 0.55
ADRB3 P13945 7/20 0.55
ADRA1D P25100 7/20 0.55
ADRA1A P35348 7/20 0.55
ADRA1B P35368 7/20 0.55
ALDH1A1 P00352 5/20 0.46
CYP2D6 P10635 3/20 0.46
MAPT P10636 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2C19 P33261 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
KDM4E B2RXH2 3/20 0.42
HSD17B10 Q99714 3/20 0.42
TSHR P16473 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
DRD3 P35462 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9501745 0.89 ADRB2 (0.55) ADRB2ADRB1ADRB3ADRA1DADRA1A
Hydrochloric Acid SCHEMBL9135234 0.88 ADRB2 (0.54) ADRB2ADRB1ADRB3ADRA1DADRA1A
SCHEMBL9703210 0.81 ALDH1A1 (0.65) ALDH1A1CYP2D6MAPTCYP1A2CYP2C19
SCHEMBL9502729 0.80 CYP24A1 (0.48) ADRB2ADRB1ADRB3ADRA1DADRA1A
SCHEMBL9504971 0.80 ALDH1A1 (0.55) ADRB2ADRB1ADRB3ADRA1AADRA1B
Hydrochloric Acid SCHEMBL9133466 0.80 CYP24A1 (0.47) ADRB2ADRB1ADRB3ADRA1DADRA1A
SCHEMBL9504939 0.79 ALDH1A1 (0.49) ADRB3ALDH1A1CYP2D6MAPTCYP1A2
Hydrochloric Acid SCHEMBL9133377 0.79 ALDH1A1 (0.48) ADRB3ALDH1A1CYP2D6MAPTCYP1A2
SCHEMBL9504910 0.78 ALDH1A1 (0.52) ADRB1ADRB3ALDH1A1CYP2D6MAPT
SCHEMBL9503443 0.78 ADRB2 (0.49) ADRB2ADRB1ADRB3ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549668-A1 ANTI-HYPERTENSIVE TETRALINS THE WELLCOME FOUNDATION LIMITED (GB) 1993-07-07 EP claimed
WO-1992005143-A1 ANTI-HYPERTENSIVE TETRALINS THE WELLCOME FOUNDATION LIMITED (GB) 1992-04-02 WO claimed