SCHEMBL9504261

SCHEMBL9504261

CCOC(=O)C1=C(C)NC(C)=C([N+](=O)[O-])C1c1cccc2c1OCCO2

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.66
AMY1A P0DUB6 1/20 0.66
GAA P10253 1/20 0.66
SI P14410 1/20 0.66
MGAM2 Q2M2H8 1/20 0.66
CACNA1C Q13936 10/20 0.52
CACNA1F O60840 7/20 0.51
CACNA1D Q01668 7/20 0.51
CACNA1S Q13698 7/20 0.51
ADORA3 P0DMS8 4/20 0.51
MAPT P10636 7/20 0.49
LMNA P02545 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP1A2 P05177 5/20 0.48
CYP3A4 P08684 5/20 0.48
CYP2C9 P11712 5/20 0.48
CYP2C19 P33261 5/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272515 0.85 MGAM (0.56) MGAMAMY1AGAASIMGAM2
SCHEMBL7272519 0.81 CACNA1C (0.53) MGAMAMY1AGAASIMGAM2
SCHEMBL9505368 0.81 GAA (0.44) MGAMAMY1AGAASIMGAM2
SCHEMBL11007622 0.80 CACNA1C (0.58) CACNA1CCACNA1FCACNA1DCACNA1SADORA3
SCHEMBL11373038 0.78 CYP2C9 (0.57) GAACACNA1CCACNA1FCACNA1DCACNA1S
SCHEMBL9518606 0.77 GAA (0.64) MGAMAMY1AGAASIMGAM2
Oxodipine SCHEMBL332244 0.76 GAA (0.91) MGAMAMY1AGAASIMGAM2
SCHEMBL11368968 0.76 CACNA1C (0.53) CACNA1CCACNA1FCACNA1DCACNA1SADORA3
SCHEMBL7265346 0.76 CYP1A2 (0.80) CACNA1CCACNA1FCACNA1DCACNA1SADORA3
SCHEMBL8680780 0.75 ADORA3 (0.67) CACNA1CCACNA1FCACNA1DCACNA1SADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
WO-1990009376-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-23 WO disclosed
EP-0383320-A1 A process for preparation of enantiomerically pure polysubstituted 1,4-dihydropyridines BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-22 EP disclosed