SCHEMBL9505368

SCHEMBL9505368

CCOC(=O)C1=C([S+](C)C(C)c2ccccc2)NC(C)=C([N+](=O)[O-])C1c1cccc2c1OCCO2.F[B-](F)(F)F.F[B-](F)(F)F.F[B-](F)(F)F.F[B-](F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.44
MGAM O43451 1/20 0.44
AMY1A P0DUB6 1/20 0.44
SI P14410 1/20 0.44
MGAM2 Q2M2H8 1/20 0.44
MAPT P10636 5/20 0.38
CACNA1C Q13936 8/20 0.36
CACNA1D Q01668 6/20 0.36
CACNA1F O60840 5/20 0.36
CACNA1S Q13698 5/20 0.36
ADORA3 P0DMS8 6/20 0.36
CYP1A2 P05177 4/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
TSHR P16473 2/20 0.36
NFKB1 P19838 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9504261 0.81 MGAM (0.66) GAAMGAMAMY1ASIMGAM2
SCHEMBL7272515 0.68 MGAM (0.56) GAAMGAMAMY1ASIMGAM2
SCHEMBL11007622 0.65 CACNA1C (0.58) MAPTCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL7272519 0.65 CACNA1C (0.53) GAAMGAMAMY1ASIMGAM2
SCHEMBL9874899 0.64 NR1I2 (0.61) GAAMAPTCACNA1CCACNA1DCACNA1F
SCHEMBL11373038 0.64 CYP2C9 (0.57) GAAMAPTCACNA1CCACNA1DCACNA1F
SCHEMBL9502266 0.63 MGAM (0.54) GAAMGAMAMY1ASIMGAM2
SCHEMBL7265346 0.63 CYP1A2 (0.80) MAPTCACNA1CCACNA1DCACNA1FCACNA1S
SCHEMBL9518606 0.63 GAA (0.64) GAAMGAMAMY1ASIMGAM2
SCHEMBL8680780 0.63 ADORA3 (0.67) MAPTCACNA1CCACNA1DCACNA1FCACNA1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
WO-1990009376-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-23 WO disclosed