SCHEMBL9507024

SCHEMBL9507024

O=C(O)c1ccc(OCCCc2ccc(O)c(O)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.53
PLA2G4B P0C869 3/20 0.52
IGF1R P08069 3/20 0.51
ALOX15 P16050 3/20 0.51
TP53 P04637 1/20 0.51
TSHR P16473 1/20 0.51
APP P05067 2/20 0.50
YWHAG P61981 1/20 0.50
LCK P06239 1/20 0.50
ALDH1A1 P00352 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
FFAR1 O14842 1/20 0.49
CYP4F2 P78329 1/20 0.48
CYP4A11 Q02928 1/20 0.48
HTT P42858 1/20 0.48
RARB P10826 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9506788 0.94 PLA2G4B (0.60) PKMPLA2G4BIGF1RALOX15TP53
SCHEMBL10412008 0.86 CYSLTR1 (0.54) PLA2G4BIGF1RALOX15APPYWHAG
SCHEMBL9558671 0.85 PLA2G4B (0.55) PKMPLA2G4BTP53TSHRALDH1A1
SCHEMBL10412747 0.84 CYSLTR1 (0.57) PLA2G4BIGF1RALOX15APPYWHAG
SCHEMBL9557988 0.83 PLA2G4B (0.57) PLA2G4BTP53TSHRHTTRARB
SCHEMBL9506806 0.81 KMT2A (0.56) PLA2G4BIGF1RALOX15
SCHEMBL7774931 0.81 PKM (0.68) PKMPLA2G4BFFAR1
SCHEMBL4361279 0.80 PLA2G4B (0.76) PKMPLA2G4BTP53TSHRFFAR1
SCHEMBL14966915 0.80 PKM (0.71) PKMPLA2G4BTP53TSHRFFAR1
SCHEMBL9507025 0.79 LCK (0.61) IGF1RALOX15APPYWHAGLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0310126-B1 DERIVATIVES OF PYROCATECHOL-CARBOXYLIC ACID, THEIR PREPARATION AND USE AS ACTIVE INGREDIENTS IN MEDICINES F. HOFFMANN-LA ROCHE AG (CH) 1993-08-18 EP disclosed
US-5191108-A Lipoxygenase inhibitors, antiinflammatory agents HOFFMANN-LA ROCHE INC. (US) 1993-03-02 US disclosed
US-5025036-A Antiinflammatory agents, gastrointestinal, cardiovascular and skin disorders HOFFMANN-LA ROCHE INC. (US) 1991-06-18 US disclosed
EP-0310126-A2 Derivatives of pyrocatechol-carboxylic acid, their preparation and use as active ingredients in medicines F. HOFFMANN-LA ROCHE AG (CH) 1989-04-05 EP disclosed