SCHEMBL9508450

SCHEMBL9508450

CC(Cl)C(=O)N1CC(C)c2ccccc2C1c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HHAT Q5VTY9 4/20 0.40
CYP2D6 P10635 1/20 0.40
NOTUM Q6P988 1/20 0.39
TACR1 P25103 1/20 0.37
TRPV1 Q8NER1 1/20 0.36
ATM Q13315 1/20 0.36
NPC1 O15118 1/20 0.36
MITF O75030 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
XBP1 P17861 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509175 0.90 NOTUM (0.40) HHATCYP2D6NOTUMTRPV1ATM
SCHEMBL9509161 0.78 HHAT (0.61) HHATCYP2D6
SCHEMBL9508210 0.74 NOTUM (0.43) NOTUMALDH1A1HTT
SCHEMBL9508465 0.73 NOTUM (0.40) HHATNOTUMALDH1A1LMNAHTT
SCHEMBL9511217 0.69 OPRD1 (0.42) NOTUMALDH1A1LMNAHTT
SCHEMBL9508172 0.68 DRD1 (0.57) HHATCYP2D6NPC1NPSR1
SCHEMBL9508456 0.67 HHAT (0.57) HHATCYP2D6
Iodide SCHEMBL27324981 0.65 MAPT (0.44) LMNA
SCHEMBL11188809 0.64 SMN1; SMN2 (0.50) ALDH1A1
SCHEMBL12153444 0.64 HHAT (0.57) HHATCYP2D6TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0230871-B1 HALOACYL 1-SUBSTITUTED-1,2,3,4-TETRAHYDROISOQUINOLINES AS HERBICIDE ANTIDOTES Monsanto Company (US) 1993-09-22 EP claimed
EP-0230871-A2 Haloacyl 1-substituted-1,2,3,4-tetrahydroisoquinolines as herbicide antidotes Monsanto Company (US) 1987-08-05 EP claimed
EP-0230871-B1 HALOACYL 1-SUBSTITUTED-1,2,3,4-TETRAHYDROISOQUINOLINES AS HERBICIDE ANTIDOTES Monsanto Company (US) 1993-09-22 EP disclosed
US-4755218-A Reducing acetochlor injury to corn by applying with antidote MONSANTO COMPANY (US) 1988-07-05 US disclosed
EP-0230871-A2 Haloacyl 1-substituted-1,2,3,4-tetrahydroisoquinolines as herbicide antidotes Monsanto Company (US) 1987-08-05 EP disclosed