SCHEMBL9508458

SCHEMBL9508458

C=CCc1cc([N+](=O)[O-])cc(N)c1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
ALDH1A1 P00352 3/20 0.44
TDP1 Q9NUW8 2/20 0.44
ALOX15 P16050 1/20 0.44
POLB P06746 3/20 0.41
HTT P42858 1/20 0.41
LMNA P02545 2/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
GPR35 Q9HC97 1/20 0.40
GAA P10253 1/20 0.37
THRB P10828 1/20 0.37
HCAR3 P49019 1/20 0.36
TP53 P04637 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10661047 0.82 HTT (0.59) CYP3A4ALDH1A1TDP1ALOX15POLB
SCHEMBL10659985 0.82 HTT (0.59) CYP3A4ALDH1A1TDP1ALOX15POLB
SCHEMBL10364596 0.82 NPC1 (0.51) ALDH1A1POLBHTTMEN1KMT2A
SCHEMBL10590043 0.80 POLB (0.51) CYP3A4ALDH1A1TDP1ALOX15POLB
SCHEMBL9695123 0.80 RAB9A (0.49) ALDH1A1TDP1POLBLMNAGAA
SCHEMBL10658167 0.78 HTT (0.50) CYP3A4ALDH1A1TDP1ALOX15POLB
SCHEMBL11757407 0.75 AKR1B1 (0.44) CYP3A4ALDH1A1TDP1ALOX15POLB
SCHEMBL1644916 0.75 CYP3A4 (0.51) CYP3A4ALDH1A1TDP1ALOX15POLB
SCHEMBL9683795 0.75 TDP1 (0.50) CYP3A4ALDH1A1TDP1ALOX15POLB
SCHEMBL17769822 0.75 ALDH1A1 (0.55) CYP3A4ALDH1A1TDP1ALOX15POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0317645-B1 4H-3,1-BENZOXAZIN-4-ONE COMPOUNDS AND SERINE PROTEASE-INHIBITING MEDICINAL COMPOSITION CONTAINING SAME TEIJIN LIMITED (JP) 1993-09-15 EP disclosed
US-4980287-A ANTIINFLAMMATORY AGENTS; INHIBITOR OF DEGENERATION AND DESTRUCTION OF TISSUES TEIJIN LIMITED (JP) 1990-12-25 US disclosed
EP-0317645-A1 4H-3,1-BENZOXAZIN-4-ONE COMPOUNDS AND SERINE PROTEASE-INHIBITING MEDICINAL COMPOSITION CONTAINING SAME TEIJIN LIMITED (JP) 1989-05-31 EP disclosed