SCHEMBL9508531

SCHEMBL9508531

COc1ccc(CSc2cc(OC)ccc2CN(C)C)cc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.51
SLC6A2 P23975 3/20 0.51
SLC6A3 Q01959 3/20 0.51
APP P05067 1/20 0.44
HTR2A P28223 1/20 0.44
KCNH2 Q12809 1/20 0.44
MAOB P27338 3/20 0.43
CYP2D6 P10635 1/20 0.42
TSHR P16473 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAOA P21397 2/20 0.41
DAO P14920 1/20 0.40
IDO1 P14902 2/20 0.40
LMNA P02545 1/20 0.39
MMP13 P45452 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509583 0.89 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3HTR2AKCNH2
SCHEMBL9507201 0.82 APP (0.46) APPMAOBCYP2D6TSHRALDH1A1
SCHEMBL10687383 0.77 APP (0.58) APPMAOBTSHRALDH1A1MAOA
SCHEMBL19297784 0.75 APP (0.49) APPMAOBCYP2D6TSHRALDH1A1
SCHEMBL15700194 0.73 SLC6A4 (0.55) SLC6A4SLC6A2SLC6A3HTR2AKCNH2
SCHEMBL9507453 0.72 IDO1 (0.45) APPMAOBCYP2D6TSHRALDH1A1
SCHEMBL9507325 0.72 MAOB (0.42) SLC6A4SLC6A2SLC6A3APPMAOB
SCHEMBL9507220 0.72 GAA (0.44) SLC6A4SLC6A2SLC6A3APPMAOB
SCHEMBL29673296 0.71 CYP1A2 (0.43) APPMAOBCYP2D6TSHRMAOA
SCHEMBL385286 0.71 HRH3 (0.58) SLC6A4SLC6A2SLC6A3TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358305-B1 MERCAPTO-PHENYLALCANOYLAMINO ACID AMIDES, THEIR PREPARATION AND THEIR USE AS COLLAGENASE INHIBITORS BEECHAM GROUP PLC (GB) 1993-08-25 EP disclosed
US-5124322-A Antiarthritic agents BEECHAM GROUP P.L.C. (GB) 1992-06-23 US disclosed
EP-0358305-A1 Mercapto-phenylalcanoylamino acid amides, their preparation and their use as collagenase inhibitors BEECHAM GROUP PLC (GB) 1990-03-14 EP disclosed