SCHEMBL9507220

SCHEMBL9507220

COc1ccc(CSc2c(CN(C)C)cccc2C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 1/20 0.44
SLC6A4 P31645 4/20 0.43
SLC6A2 P23975 3/20 0.43
SLC6A3 Q01959 3/20 0.43
FABP3 P05413 1/20 0.39
FABP4 P15090 1/20 0.39
APP P05067 1/20 0.38
MAOB P27338 3/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TSHR P16473 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509595 0.85 GAA (0.41) GAAKMT2AMEN1ALDH1A1FABP3
SCHEMBL9510979 0.74 MMP1 (0.42) GAAKMT2AMEN1ALDH1A1MAPT
SCHEMBL9508531 0.72 SLC6A4 (0.51) ALDH1A1SLC6A4SLC6A2SLC6A3APP
SCHEMBL9507496 0.71 HTR7 (0.46) KMT2AMEN1ALDH1A1SLC6A4SLC6A2
SCHEMBL9509583 0.68 SLC6A4 (0.44) KMT2AMEN1SLC6A4SLC6A2SLC6A3
SCHEMBL9507325 0.68 MAOB (0.42) KMT2AMEN1ALDH1A1SLC6A4SLC6A2
SCHEMBL10705108 0.67 GAA (0.58) GAAKMT2AMEN1ALDH1A1MAOB
SCHEMBL12831776 0.67 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3CYP3A4CYP2D6
SCHEMBL30716088 0.65 TP53 (0.46) GAAKMT2AMEN1FABP3FABP4
SCHEMBL31075610 0.65 FABP3 (0.43) FABP3FABP4APPMAOBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358305-B1 MERCAPTO-PHENYLALCANOYLAMINO ACID AMIDES, THEIR PREPARATION AND THEIR USE AS COLLAGENASE INHIBITORS BEECHAM GROUP PLC (GB) 1993-08-25 EP disclosed
US-5124322-A Antiarthritic agents BEECHAM GROUP P.L.C. (GB) 1992-06-23 US disclosed
EP-0358305-A1 Mercapto-phenylalcanoylamino acid amides, their preparation and their use as collagenase inhibitors BEECHAM GROUP PLC (GB) 1990-03-14 EP disclosed