SCHEMBL9508752

SCHEMBL9508752

CCc1ccc(-c2ccc(C#Cc3ccc(C)cc3)c(F)c2F)cc1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 8/20 0.37
CYP2A6 P11509 1/20 0.35
KCNH2 Q12809 3/20 0.34
ACACB O00763 3/20 0.33
KDM1A O60341 1/20 0.33
CA12 O43570 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
GRM5 P41594 1/20 0.33
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RARG P13631 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509130 1.00 FFAR1 (0.37) FFAR1CYP2A6KCNH2ACACBKDM1A
SCHEMBL9511355 0.94 CYP2A6 (0.39) FFAR1CYP2A6ACACBRARARARB
SCHEMBL9508754 0.90 LMNA (0.40) FFAR1CYP2A6ACACBGRM5RARA
SCHEMBL9510036 0.89 GRM5 (0.39) FFAR1CYP2A6KCNH2CA12CA2
SCHEMBL9512412 0.89 FFAR1 (0.41) FFAR1ACACB
SCHEMBL9512352 0.89 FFAR1 (0.41) FFAR1ACACB
SCHEMBL9512399 0.87 FFAR1 (0.36) FFAR1CYP2A6ACACBKDM1ARARB
SCHEMBL9509318 0.87 FFAR1 (0.36) FFAR1CYP2A6ACACBKDM1ARARB
SCHEMBL10511143 0.87 TSHR (0.40) FFAR1RARARARBRARG
SCHEMBL10512751 0.87 TSHR (0.40) FFAR1RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308438-B1 LIQUID CRYSTAL PHASE CONTAINING TOLANES MERCK PATENT GmbH (DE) 1993-09-29 EP disclosed