SCHEMBL9508754

SCHEMBL9508754

CCc1ccc(-c2ccc(C#Cc3ccc(F)cc3)c(F)c2F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
GCGR P47871 1/20 0.39
MAPK14 Q16539 1/20 0.39
FFAR1 O14842 3/20 0.38
CYP2A6 P11509 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GRM5 P41594 2/20 0.35
ACACB O00763 2/20 0.34
ADCY1 Q08828 1/20 0.34
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RARG P13631 1/20 0.32
GAA P10253 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
NPC1 O15118 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAOA P21397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9511355 0.95 CYP2A6 (0.39) LMNAGCGRMAPK14FFAR1CYP2A6
SCHEMBL9509130 0.90 FFAR1 (0.37) FFAR1CYP2A6GRM5ACACBRARA
SCHEMBL9508752 0.90 FFAR1 (0.37) FFAR1CYP2A6GRM5ACACBRARA
SCHEMBL9512399 0.89 FFAR1 (0.36) FFAR1CYP2A6ACACBRARB
SCHEMBL9512281 0.89 FFAR1 (0.42) LMNAFFAR1GRM5ACACBGAA
SCHEMBL9509318 0.89 FFAR1 (0.36) FFAR1CYP2A6ACACBRARB
SCHEMBL9510180 0.86 TSHR (0.40) FFAR1RARB
SCHEMBL9509936 0.86 FFAR1 (0.40) FFAR1RARBGAAKMT2AHTT
SCHEMBL9511464 0.86 TSHR (0.40) FFAR1RARB
SCHEMBL9510169 0.85 TSHR (0.46) FFAR1RARARARBRARGMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308438-B1 LIQUID CRYSTAL PHASE CONTAINING TOLANES MERCK PATENT GmbH (DE) 1993-09-29 EP disclosed