SCHEMBL9511642

SCHEMBL9511642

CCOC(=O)CCCC1(CCCC(=O)OCC)CC(=O)c2ccc(O)cc2O1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.50
ALDH1A1 P00352 5/20 0.50
KMT2A Q03164 1/20 0.46
HPGD P15428 4/20 0.42
GAA P10253 3/20 0.42
CASP1 P29466 3/20 0.42
HSD17B10 Q99714 3/20 0.42
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
BRD4 O60885 1/20 0.39
HTR2C P28335 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9635631 0.83 KDM4E (0.54) KDM4EALDH1A1KMT2AHPGDGAA
SCHEMBL3029269 0.78 ALDH1A1 (0.66) KDM4EALDH1A1KMT2AHTR2CMAPT
SCHEMBL9512184 0.77 KDM4E (0.46) KDM4EALDH1A1HPGDGAACASP1
SCHEMBL10639092 0.74 AKT1 (0.60) KDM4EALDH1A1KMT2AHPGDGAA
SCHEMBL30065886 0.73 ALDH1A1 (0.61) KDM4EALDH1A1KMT2AHTR2CMAPT
SCHEMBL10638595 0.71 KDM4E (0.39) KDM4EALDH1A1KMT2AHPGDGAA
SCHEMBL10695261 0.70 BRD4 (0.50) KDM4EALDH1A1HPGDGAACASP1
SCHEMBL11369382 0.69 KDM4E (0.68) KDM4EALDH1A1KMT2AHTR2CMAPT
SCHEMBL10344387 0.69 BRD4 (0.49) KDM4EALDH1A1HPGDGAACASP1
SCHEMBL11112069 0.68 KDM4E (0.59) KDM4EALDH1A1HTR2CMAPTAKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0342664-B1 2,2-disubstituted benzopyran leukotriene-D4 antagonists SEARLE & CO (US) 1993-12-15 EP disclosed
US-5093353-A 2,2-di-substituted benzopyran leukotriene-D4 antagonists G. D. SEARLE & CO. (US) 1992-03-03 US disclosed
EP-0342664-A2 2,2-disubstituted benzopyran leukotriene-D4 antagonists G.D. Searle & Co. (US) 1989-11-23 EP disclosed